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<p>Understanding the Glycopeptide Antibiotic Crosslinking Cascade: In Vitro Approaches Reveal the Details of a Complex Biosynthesis Pathway.<em> ChemBioChem</em> (2020) 22, 43-51.</p>
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<p>Synthesis of the C1-C27 Fragment of Stambomycin D Validates Modular Polyketide Synthase-Based Stereochemical Assignments.<em> Organic Letters</em> (2021) 23, 7439-7444.</p>
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<p>A Bimodal Fluorescence-Raman Probe for Cellular Imaging.<em> Cells</em> (2021) 10, 1699.</p>
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<p>An Ultrapotent and Selective Cyclic Peptide Inhibitor of Human β-Factor XIIa in a Cyclotide Scaffold.<em> Journal of the American Chemical Society</em> (2021) 143, 18481-18489.</p>
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<p>Synthesis of 13C/19F/2H Labeled Indoles for Use as Tryptophan Precursors for Protein NMR Spectroscopy.<em> Organic & Biomolecular Chemistry</em> (2021) 19, 5133-5147.</p>
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<p>A Versatile Fluorescent Sensor Array for Platinum Anticancer Drug Detection in Biological Fluids.<em> ACS Sensors</em> (2021) 6, 1261-1269.</p>
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<p>Antimicrobial and Anticancer Properties of Synthetic Peptides Derived from the Wasp Parachartergus Fraternus.<em> ChemBioChem</em> (2021) 22, 1415-1423.</p>
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<p>Discovery of the Pseudomonas Polyyne Protegencin by a Phylogeny-Guided Study of Polyyne Biosynthetic Gene Cluster Diversity.<em> mBio</em> (2021) 12</p>
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<p>Design of a Stable Cyclic Peptide Analgesic Derived from Sunflower Seeds That Targets the κ-Opioid Receptor for the Treatment of Chronic Abdominal Pain.<em> Journal of Medicinal Chemistry</em> (2021) 64, 9042-9055.</p>
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<p>Designed β-Hairpins Inhibit LDH5 Oligomerization and Enzymatic Activity.<em> Journal of Medicinal Chemistry</em> (2021) 64, 3767-3779.</p>
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<p>Multipurpose Peptides: The Venoms of Amazonian Stinging Ants Contain Anthelmintic Ponericins with Diverse Predatory and Defensive Activities.<em> Biochemical Pharmacology</em> (2021) 192, 114693.</p>
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<p>Discovery of Cyclic Peptide Ligands to the SARS-CoV-2 Spike Protein Using mRNA Display.<em> ACS Central Science</em> (2021) 7, 1001-1008.</p>
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<p>Proteome Analysis and Epitope Mapping in a Commercial Reduced-Gluten Wheat Product.<em> Frontiers in Nutrition</em> (2021) 8</p>
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<p>Through-Space Scalar 19F-19F Couplings between Fluorinated Noncanonical Amino Acids for the Detection of Specific Contacts in Proteins.<em> Journal of the American Chemical Society</em> (2021) 143, 19587-19598.</p>
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<p>BET-Family Bromodomains Can Recognize Diacetylated Sequences from Transcription Factors Using a Conserved Mechanism.<em> Biochemistry</em> (2021) 60, 648-662.</p>
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<p class="jp-name">Tran, H. N. T.; Tran, P.; Deuis, J. R.; McMahon, K. L.; Yap, K.; Craik, D. J.; Vetter, I.; Schroeder, C. I.</p>
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<p class="jp-name">Ullrich, S.; Sasi, V. M.; Mahawaththa, M. C.; Ekanayake, K. B.; Morewood, R.; George, J.; Shuttleworth, L.; Zhang, X.; Whitefield, C.; Otting, G.; Jackson, C.; Nitsche, C.</p>
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<p>Sunflower Trypsin Inhibitor-1 (SFTI-1): Sowing Seeds in the Fields of Chemistry and Biology.<em> Angewandte Chemie International Edition</em> (2020) 60, 8050-8071.</p>
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<p class="jp-name">Chen, K.-E.; Guo, Q.; Hill, T. A.; Cui, Y.; Kendall, A. K.; Yang, Z.; Hall, R. J.; Healy, M. D.; Sacharz, J.; Norwood, S. J.; Fonseka, S.; Xie, B.; Reid, R. C.; Leneva, N.; Parton, R. G.; Ghai, R.; Stroud, D. A.; Fairlie, D. P.; Suga, H.; Jackson, L. P.; Teasdale, R. D.; Passioura, T.; Collins, B. M.</p>
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<p>De Novo Macrocyclic Peptides for Inhibiting, Stabilizing, and Probing the Function of the Retromer Endosomal Trafficking Complex.<em> Science Advances</em> (2021) 7</p>
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<p>The Evolution and Engineering of Enzyme Activity through Tuning Conformational Landscapes.<em> Protein Engineering, Design and Selection</em> (2021) 34</p>
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<p>In Planta Discovery and Chemical Synthesis of Bracelet Cystine Knot Peptides from Rinorea Bengalensis.<em> Journal of Natural Products</em> (2021) 84, 395-407.</p>
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<p class="jp-name">Depuydt, A.-S.; Rihon, J.; Cheneval, O.; Vanmeert, M.; Schroeder, C. I.; Craik, D. J.; Lescrinier, E.; Peigneur, S.; Tytgat, J.</p>
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<p>Cyclic Peptides as T-Type Calcium Channel Blockers: Characterization and Molecular Mapping of the Binding Site.<em> ACS Pharmacology & Translational Science</em> (2021) 4, 1379-1389.</p>
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<p>Synthesis and Evaluation of Peptidic Thrombin Inhibitors Bearing Acid-Stable Sulfotyrosine Analogues.<em> Chemical Communications</em> (2021) 57, 10923-10926.</p>
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<p>Total Synthesis of the Spider-Venom Peptide Hi1a.<em> Organic Letters</em> (2021) 23, 8375-8379.</p>
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<p>Melanocortin 1 Receptor Agonists Based on a Bivalent, Bicyclic Peptide Framework.<em> Journal of Medicinal Chemistry</em> (2021) 64, 9906-9915.</p>
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<p>Perennial Ryegrass Contains Gluten-Like Proteins That Could Contaminate Cereal Crops.<em> Frontiers in Nutrition</em> (2021) 8</p>
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<p class="jp-name">Fage, C. D.; Kosol, S.; Jenner, M.; öster, C.; Gallo, A.; Kaniusaite, M.; Steinbach, R.; Staniforth, M.; Stavros, V. G.; Marahiel, M. A.; Cryle, M. J.; Lewandowski, J. R.</p>
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<p>Communication Breakdown: Dissecting the COM Interfaces between the Subunits of Nonribosomal Peptide Synthetases.<em> ACS Catalysis</em> (2021) 11, 10802-10813.</p>
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<p class="jp-name">Ford, D. J.; Duggan, N. M.; Fry, S. E.; Ripoll-Rozada, J.; Agten, S. M.; Liu, W.; Corcilius, L.; Hackeng, T. M.; van Oerle, R.; Spronk, H. M. H.; Ashhurst, A. S.; Mini Sasi, V.; Kaczmarski, J. A.; Jackson, C. J.; Pereira, P. J. B.; Passioura, T.; Suga, H.; Payne, R. J.</p>
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<p>Potent Cyclic Peptide Inhibitors of FXIIa Discovered by mRNA Display with Genetic Code Reprogramming.<em> Journal of Medicinal Chemistry</em> (2021) 64, 7853-7876.</p>
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<p>Acid-Sensing Ion Channels: Expression and Function in Resident and Infiltrating Immune Cells in the Central Nervous System.<em> Frontiers in Cellular Neuroscience</em> (2021) 15</p>
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<p>Substrate Dynamics Contribute to Enzymatic Specificity in Human and Bacterial Methionine Adenosyltransferases.<em> JACS Au</em> (2021) 1, 2349-2360.</p>
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<p>Tuning the Anti-Angiogenic Effect of the P15 Peptide Using Cyclic Trypsin Inhibitor Scaffolds.<em> ACS Chemical Biology</em> (2021) 16, 829-837.</p>
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<p>Sulfotyrosine-Mediated Recognition of Human Thrombin by a Tsetse Fly Anticoagulant Mimics Physiological Substrates.<em> Cell Chemical Biology</em> (2021) 28, 26-33.e8.</p>
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<p>Late-Stage Modification of Peptides and Proteins at Cysteine with Diaryliodonium Salts.<em> Chemical Science</em> (2021) 12, 14159-14166.</p>
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<p>Proteome and Nutritional Shifts Observed in Hordein Double-Mutant Barley Lines.<em> Frontiers in Plant Science</em> (2021) 12</p>
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<p>Protein Extraction Protocols for Optimal Proteome Measurement and Arginine Kinase Quantitation from Cricket Acheta Domesticus for Food Safety Assessment.<em> Food Chemistry</em> (2021) 348, 129110.</p>
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<p class="jp-name">Benfield, A. H.; Defaus, S.; Lawrence, N.; Chaousis, S.; Condon, N.; Cheneval, O.; Huang, Y.-H.; Chan, L. Y.; Andreu, D.; Craik, D. J.; Henriques, S. T.</p>
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<p>Cyclic Gomesin, a Stable Redesigned Spider Peptide Able to Enter Cancer Cells.<em> Biochimica et Biophysica Acta (BBA) - Biomembranes</em> (2021) 1863, 183480.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1016/j.bbamem.2020.183480" target="_blank">10.1016/j.bbamem.2020.183480</a></div>
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<p class="jp-name">Ashwood, L. M.; Mitchell, M. L.; Madio, B.; Hurwood, D. A.; King, G. F.; Undheim, E. A. B.; Norton, R. S.; Prentis, P. J.</p>
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<p>Tentacle Morphological Variation Coincides with Differential Expression of Toxins in Sea Anemones.<em> Toxins</em> (2021) 13, 452.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.3390/toxins13070452" target="_blank">10.3390/toxins13070452</a></div>
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<p class="jp-name">Araujo, A. D.; Nguyen, H. T.; Fairlie, D. P.</p>
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<p>Late-Stage Hydrocarbon Conjugation and Cyclisation in Synthetic Peptides and Proteins.<em> ChemBioChem</em> (2021) 22, 1784-1789.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1002/cbic.202000796" target="_blank">10.1002/cbic.202000796</a></div>
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<p class="jp-name">Aragaw, W. W.; Lee, B. M.; Yang, X.; Zimmerman, M. D.; Gengenbacher, M.; Dartois, V.; Chui, W.-K.; Jackson, C. J.; Dick, T.</p>
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<p>Potency Boost of a Mycobacterium Tuberculosis Dihydrofolate Reductase Inhibitor by Multienzyme F 420 H 2 -Dependent Reduction.<em> Proceedings of the National Academy of Sciences</em> (2021) 118</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1073/pnas.2025172118" target="_blank">10.1073/pnas.2025172118</a></div>
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<p class="jp-name">Agten, S. M.; Watson, E. E.; Ripoll-Rozada, J.; Dowman, L. J.; Wu, M. C. L.; Alwis, I.; Jackson, S. P.; Pereira, P. J. B.; Payne, R. J.</p>
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<p>Potent Trivalent Inhibitors of Thrombin through Hybridization of Salivary Sulfopeptides from Hematophagous Arthropods.<em> Angewandte Chemie International Edition</em> (2021) 60, 5348-5356.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1002/anie.202015127" target="_blank">10.1002/anie.202015127</a></div>
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<p class="jp-name">Abdelkader, E. H.; Qianzhu, H.; Tan, Y. J.; Adams, L. A.; Huber, T.; Otting, G.</p>
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<p>Genetic Encoding of N6-(((Trimethylsilyl)Methoxy)Carbonyl)-l-Lysine for NMR Studies of Protein-Protein and Protein-Ligand Interactions.<em> Journal of the American Chemical Society</em> (2021) 143, 1133-1143.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1021/jacs.0c11971" target="_blank">10.1021/jacs.0c11971</a></div>
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<p class="jp-name">Abdelkader, E. H.; Otting, G.</p>
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<p>NT*-HRV3CP: An Optimized Construct of Human Rhinovirus 14 3C Protease for High-Yield Expression and Fast Affinity-Tag Cleavage.<em> Journal of Biotechnology</em> (2021) 325, 145-151.</p>
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<div class="journal-papers-doi"><span>DOI:</span> <a href="https://doi.org/10.1016/j.jbiotec.2020.11.005" target="_blank">10.1016/j.jbiotec.2020.11.005</a></div>
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